BDBM220664 US10633379, Compound Y::US9296741, 253
SMILES CCNC(=O)c1cc2c(cn(C)c(=O)c2[nH]1)-c1cc(ccc1Oc1ccc(F)cc1F)S(C)(=O)=O
InChI Key InChIKey=GLPRVXBSUHOVMP-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 220664
Affinity DataKi: 1.20nMAssay Description:Binding affinity to BDR4- BD2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human N-terminal His6 tagged BRD4 BD2 (352 to 457) residues expressed in Escherichia coli BL21(DE3) cells after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of human N-terminal His6 tagged BRD4 BD1 (57 to 168) residues expressed in Escherichia coli BL21(DE3) cells after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity to BDR4-BD1 (unknown origin)More data for this Ligand-Target Pair