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Found 4 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM220664'
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM220664(US10633379, Compound Y | US9296741, 253)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to BDR4- BD2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM220664(US10633379, Compound Y | US9296741, 253)
Affinity DataKi:  1.30nMAssay Description:Inhibition of human N-terminal His6 tagged BRD4 BD2 (352 to 457) residues expressed in Escherichia coli BL21(DE3) cells after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM220664(US10633379, Compound Y | US9296741, 253)
Affinity DataKi:  22nMAssay Description:Binding affinity to BDR4-BD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM220664(US10633379, Compound Y | US9296741, 253)
Affinity DataKi:  22nMAssay Description:Inhibition of human N-terminal His6 tagged BRD4 BD1 (57 to 168) residues expressed in Escherichia coli BL21(DE3) cells after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB