BDBM50652109 Pimicotinib::ABSK-021 FREE BASE ANHYDROUS::ABSK-021-0 FREE BASE ANHYDROUS::ABSK-021-7::ABSK021 FREE BASE ANHYDROUS::ABSK021-NX::ASYM-133040

SMILES Cc1nc(NC(=O)N2CCC(C)(C)C2=O)ccc1Oc1ccnc(-c2cnn(C)c2)c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50652109   

TargetMacrophage colony-stimulating factor 1 receptor(Human)
University of Sharjah

Curated by ChEMBL
LigandPNGBDBM50652109(Pimicotinib | ABSK-021 FREE BASE ANHYDROUS | ABSK-...)
Affinity DataIC50: 19nMAssay Description:Inhibition of CSF1R (unknown origin) using ATP as substrate incubated for 1 hr by Z-LYTE based FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
University of Sharjah

Curated by ChEMBL
LigandPNGBDBM50652109(Pimicotinib | ABSK-021 FREE BASE ANHYDROUS | ABSK-...)
Affinity DataIC50: 77nMAssay Description:Inhibition of KIT (unknown origin) preincubated for 60 mins followed by ATP addition and measured after 1 hr by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
University of Sharjah

Curated by ChEMBL
LigandPNGBDBM50652109(Pimicotinib | ABSK-021 FREE BASE ANHYDROUS | ABSK-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of PDGFRalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed