BDBM50278350 4-fluoro-1-(4-(3-(piperidin-1-yl)propoxy)benzyl)piperidine::CHEMBL2203701::CHEMBL513193
SMILES FC1CCN(Cc2ccc(OCCCN3CCCCC3)cc2)CC1
InChI Key InChIKey=DGVKMLVLUHANCZ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50278350
Affinity DataKi: 0.0933nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant human histamine H3 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0940nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant human histamine H3 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0940nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.340nMAssay Description:Binding affinity to rat brain histamine H3 receptor after 1 hr by gamma countingMore data for this Ligand-Target Pair
Affinity DataKd: >3.00E+3nMAssay Description:Binding affinity to rat histamine H3 receptor low affinity site after 1 hr by Schard plot analysisMore data for this Ligand-Target Pair