BDBM50532781 CHEMBL4571241

SMILES CCc1ccc2n(C)c(C)c(C(=O)Nc3ccc(Oc4ncnc5cc(OC)c(OC)cc45)c(F)c3)c(=O)c2c1

InChI Key InChIKey=IKENQUDOTQBCJH-UHFFFAOYSA-N

Data  12 IC50  34 Kd

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 46 hits for monomerid = 50532781   

TargetSTE20-like serine/threonine-protein kinase(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  240nMAssay Description:Binding affinity to human SLKMore data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetMast/stem cell growth factor receptor Kit(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  1.67E+3nMAssay Description:Binding affinity to human KITMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  4nMAssay Description:Binding affinity to human FLT3More data for this Ligand-Target Pair

Target InfoPDBNCI pathwayReactome pathway
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetALK tyrosine kinase receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human ALKMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetHigh affinity nerve growth factor receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  50nMAssay Description:Binding affinity to human TRKAMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathway
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetTyrosine-protein kinase receptor TYRO3(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  58nMAssay Description:Binding affinity to human Tyro3More data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetHigh affinity nerve growth factor receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  50nMAssay Description:Binding affinity to human TRKAMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathway
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetDual specificity mitogen-activated protein kinase kinase 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  38nMAssay Description:Binding affinity to human MEK5More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetSerine/threonine-protein kinase 10(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  10nMAssay Description:Binding affinity to human LOKMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetHomeodomain-interacting protein kinase 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  11nMAssay Description:Binding affinity to human HIPk4More data for this Ligand-Target Pair

Target InfoKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  4nMAssay Description:Binding affinity to human FLT3More data for this Ligand-Target Pair

Target InfoPDBNCI pathwayReactome pathway
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetCyclin-dependent kinase 11B(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  470nMAssay Description:Binding affinity to human CDK11More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetAurora kinase B(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50:  114nMAssay Description:Inhibition of aurora B (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetTyrosine-protein kinase Blk(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  200nMAssay Description:Binding affinity to human BLKMore data for this Ligand-Target Pair

Target InfoReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetALK tyrosine kinase receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human ALKMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  2.70nMAssay Description:Binding affinity to human AXL by active site dependent completion binding assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetBDNF/NT-3 growth factors receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  54nMAssay Description:Binding affinity to human TRKBMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetSTE20-like serine/threonine-protein kinase(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  240nMAssay Description:Binding affinity to human SLKMore data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetTyrosine-protein kinase Mer(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  1.40nMAssay Description:Binding affinity to human MERMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetDual specificity mitogen-activated protein kinase kinase 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  38nMAssay Description:Binding affinity to human MEK5More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetSerine/threonine-protein kinase 10(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  10nMAssay Description:Binding affinity to human LOKMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50: <10nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBNCI pathwayReactome pathway
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetDiscoidin domain-containing receptor 2(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50:  350nMAssay Description:Inhibition of DDR2 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProtUniProtKB/TrEMBL
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetCyclin-dependent kinase 11B(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  470nMAssay Description:Binding affinity to human CDK11More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetAurora kinase A(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50:  192nMAssay Description:Inhibition of aurora A (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetTyrosine-protein kinase Blk(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  200nMAssay Description:Binding affinity to human BLKMore data for this Ligand-Target Pair

Target InfoReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  2.70nMAssay Description:Binding affinity to human AXL by active site dependent completion binding assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetHepatocyte growth factor receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  79nMAssay Description:Binding affinity to human METMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProtUniProtKB/TrEMBL
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetMast/stem cell growth factor receptor Kit(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  1.67E+3nMAssay Description:Binding affinity to human KITMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetEpithelial discoidin domain-containing receptor 1(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50:  22nMAssay Description:Inhibition of DDR1 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProtUniProtKB/TrEMBL
B.MOADDrugBankGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  2.70nMAssay Description:Binding affinity to human AXLMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant AXL incubated for 1 to 1.5 hrs by FRET based Z'-Lyte kinase assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetTyrosine-protein kinase Mer(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  1.40nMAssay Description:Binding affinity to human MERMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetBDNF/NT-3 growth factors receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  54nMAssay Description:Binding affinity to human TRKBMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50: <10nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBNCI pathwayReactome pathway
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetAurora kinase A(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50:  192nMAssay Description:Inhibition of aurora A (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetTyrosine-protein kinase receptor TYRO3(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  58nMAssay Description:Binding affinity to human Tyro3More data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetAurora kinase B(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50:  114nMAssay Description:Inhibition of aurora B (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetCyclin-dependent kinase 8(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human CDK8More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetHepatocyte growth factor receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  79nMAssay Description:Binding affinity to human METMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProtUniProtKB/TrEMBL
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetHomeodomain-interacting protein kinase 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  11nMAssay Description:Binding affinity to human HIPk4More data for this Ligand-Target Pair

Target InfoKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetEpithelial discoidin domain-containing receptor 1(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50:  22nMAssay Description:Inhibition of DDR1 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProtUniProtKB/TrEMBL
B.MOADDrugBankGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd:  2.70nMAssay Description:Binding affinity to human AXLMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant AXL incubated for 1 to 1.5 hrs by FRET based Z'-Lyte kinase assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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TargetCyclin-dependent kinase 8(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human CDK8More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetDiscoidin domain-containing receptor 2(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50532781(CHEMBL4571241)Copy SMILESCopy InChI

Affinity DataIC50:  350nMAssay Description:Inhibition of DDR2 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProtUniProtKB/TrEMBL
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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