BDBM60579 (5Z)-5-(4-hydroxybenzylidene)thiazolidine-2,4-quinone::(5Z)-5-[(4-hydroxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione::(5Z)-5-[(4-hydroxyphenyl)methylidene]thiazolidine-2,4-dione::MLS000680460::SMR000324608::cid_1276529
SMILES Oc1ccc(\C=C2/SC(=O)NC2=O)cc1
InChI Key InChIKey=ARHIHDVVUHVQCP-YVMONPNESA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 60579
Affinity DataKi: 374nMAssay Description:Competitive inhibition of mushroom tyrosinase using L-tyrosine as substrate at 1.25 uM by Line-Weaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Competitive inhibition of mushroom tyrosinase using L-tyrosine as substrate at 20 uM by Line-Weaver-Burk plot analysisMore data for this Ligand-Target Pair
Target15-hydroxyprostaglandin dehydrogenase [NAD(+)](Human)
Industry-Academic Cooperation Foundation, Chosun University
US Patent
Industry-Academic Cooperation Foundation, Chosun University
US Patent
Affinity DataIC50: 1.01E+4nMpH: 7.5Assay Description:Experimental was performed by measuring the formation of NADH at 340 nm with a fluorescence spectrophotometer. Specifically, 2 ml (in total) of the s...More data for this Ligand-Target Pair
Affinity DataIC50: 8.96E+3nMAssay Description:Inhibition of aldose reductaseMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Human)
Alma Mater Studiorum-University of Bologna
Curated by ChEMBL
Alma Mater Studiorum-University of Bologna
Curated by ChEMBL
Affinity DataIC50: 8.99E+3nMAssay Description:Inhibition of GSK3beta (unknown origin) using GS-2 peptide substrate incubated for 30 mins by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.01E+4nMAssay Description:Inhibition of aldose reductase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of mushroom tyrosinase activity using L-tyrosine as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.02E+4nMAssay Description:Inhibition of aldose reductase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.24E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair