BDBM690108 N-(5-(5-cyclopropyl-2H-tetrazol-2-yl)-2-methylphenyl)-5-(1-(2-hydroxyethyl)-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyridine-3-carboxamide::US20240262826, Compound 52

SMILES Cc1ccc(cc1NC(=O)c1cnn2ccc(cc12)-c1cnn(CCO)c1)-n1nnc(n1)C1CC1

InChI Key InChIKey=BWFLRPMLJOKIEZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 690108   

TargetMast/stem cell growth factor receptor Kit(Human)
Blueprint Medicines

US Patent
LigandPNGBDBM690108(N-(5-(5-cyclopropyl-2H-tetrazol-2-yl)-2-methylphen...)
Affinity DataIC50: 0.700nMAssay Description:For the PathScan phospho c-kit (Tyr719) sandwich ELISA: M-07e cells were resuspended at 2×106 cells/mL in phenol red free, serum-free, GM-CSF-free Is...More data for this Ligand-Target Pair
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Date in BDB:
11/25/2024
Entry Details
US Patent