BDBM808013 N-[4-(2-{M-[2-(4-Acryloyl-2-Oxo-1-Piperazinyl)Ethyl]Phenylamino}-4-Pyrimidinyloxy)-3-Fluorophenyl]-1-(P-Fluorophenyl)-5-(Trifluoromethyl)-4-Pyrazolecarboxamide ::US20260132158, Example 47

SMILES CCCN1CCN(CCc2cccc(Nc3nccc(Oc4ccc(NC(=O)c5cnn(-c6ccc(F)cc6)c5C(F)(F)F)cc4F)n3)c2)CC1

InChI Key InChIKey=FSTDXNHRPKZKRW-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 808013   

TargetMacrophage-stimulating protein receptor(Human)
The Translational Genomics Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 808013BDBM808013(N-[4-(2-{M-[2-(4-Acryloyl-2-Oxo-1-Piperazinyl)Ethy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Kinase assay was done by following instructions from the kit. Briefly, a ten-point serial dilution of compound was prepared at 5× in assay buffer wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/23/2026
Entry Details
US Patent

TargetHepatocyte growth factor receptor(Human)
The Translational Genomics Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 808013BDBM808013(N-[4-(2-{M-[2-(4-Acryloyl-2-Oxo-1-Piperazinyl)Ethy...)
Affinity DataIC50: 3.00E+3nMAssay Description:Kinase assay was done by following instructions from the kit. Briefly, a ten point serial dilution of compound was prepared at 5× in assay buffer wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/23/2026
Entry Details
US Patent