BDBM225901 MAP19::US9855269, Compound 342

SMILES Cc1c[nH]nc1-c1cccc(-c2ccc3ncnc(N)c3n2)c1

InChI Key InChIKey=COKPJYACYSCAQR-UHFFFAOYSA-N

Data  1 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 225901   

LigandChemical structure of BindingDB Monomer ID 225901BDBM225901(MAP19 | US9855269, Compound 342)
Affinity DataIC50: 3.11nMAssay Description:The kinase activity of purified human MAP4K4 kinase domain was measured by monitoring the phosphorylation of a peptide substrate derived from moesin ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 225901BDBM225901(MAP19 | US9855269, Compound 342)
Affinity DataKi:  3.66nM IC50: 3.11nMAssay Description:Z'Lyte AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2017
Entry Details
D3R