BDBM121261 US8722896, (-)-(3R)-1-(N-methyl-indol-4- ylmethyl)-N-(9-chloro-3,4- dihydro-2H-1,5-benzodioxepin- 7-ylmethyl)-N- isobutylpiperidine-3- carboxamide
SMILES CC(C)CN(Cc1cc(Cl)c2OCCCOc2c1)C(=O)C1CCCN(Cc2cccc3n(C)ccc23)C1
InChI Key InChIKey=OQQYUUDNHQHZFJ-UHFFFAOYSA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 121261
TargetProkineticin receptor 2(Cricetulus griseus (Chinese hamster))
The Regents of The University of California
US Patent
The Regents of The University of California
US Patent
Affinity DataKi: 1.24nM ΔG°: -12.6kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents of The University of California
US Patent
The Regents of The University of California
US Patent
Affinity DataKi: 3.74nM ΔG°: -12.0kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents of The University of California
US Patent
The Regents of The University of California
US Patent
Affinity DataKi: 4.26nM ΔG°: -11.9kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair