BDBM121294 US8722896, (-)-(3R)-1-(Indol-7-ylmethyl)-N- (9-chloro-2,3,4,5-tetrahydro-1- benzoxepin-7-ylmethyl)-N- isobutylpiperidine-3- carboxamide
SMILES CC(C)CN(Cc1cc(Cl)c2OCCCCc2c1)C(=O)C1CCCN(Cc2cccc3cc[nH]c23)C1
InChI Key InChIKey=WSFCSRFSULFQNX-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 121294
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents of The University of California
US Patent
The Regents of The University of California
US Patent
Affinity DataKi: 3.68nM ΔG°: -12.0kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
TargetProkineticin receptor 2(Cricetulus griseus (Chinese hamster))
The Regents of The University of California
US Patent
The Regents of The University of California
US Patent
Affinity DataKi: 7nM ΔG°: -11.6kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair