BDBM14158 APC-11922::CHEMBL293260::N-(4-carbamimidoyl-3-fluorophenyl)-2-hydroxy-3-iodo-5-methylbenzamide
SMILES Cc1cc(I)c(O)c(c1)C(=O)Nc1ccc(C(N)=N)c(F)c1
InChI Key InChIKey=GDPHNLIBJUAUNC-UHFFFAOYSA-N
Data 11 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 11 hits for monomerid = 14158
Affinity DataKi: 270nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
Affinity DataKi: 270nM ΔG°: -8.86kcal/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Inhibition of coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Activation of plasminogenMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair