BDBM14230 5-(carboxymethoxy)-3,7-dithiatricyclo[6.4.0.0^{2,6}]dodeca-1(8),2(6),4,9,11-pentaene-4-carboxylic acid::thienobenzothiophene 20
SMILES OC(=O)COc1c(sc2c1sc1ccccc21)C(O)=O
InChI Key InChIKey=NGSARUJAKPRRDR-UHFFFAOYSA-N
Data 6 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 14230
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 4.10E+3nMAssay Description:Inhibition of PTPN1More data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nM ΔG°: -7.34kcal/moleT: 2°CAssay Description:The enzymatic assay was carried out at room temperature in 96-well plates. The initial rate of PTPase-catalyzed hydrolysis of p-nitrophenol phosphate...More data for this Ligand-Target Pair
Affinity DataKi: 9.20E+3nMAssay Description:Inhibition of PTPN2More data for this Ligand-Target Pair
Affinity DataKi: 9.20E+3nM ΔG°: -6.87kcal/moleT: 2°CAssay Description:The enzymatic assay was carried out at room temperature in 96-well plates. The initial rate of PTPase-catalyzed hydrolysis of p-nitrophenol phosphate...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 1.10E+6nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: >1.25E+6nMAssay Description:Inhibition of PTPRCMore data for this Ligand-Target Pair