BDBM143693 US9682959, 1::US9751856, 1
SMILES CN1C(=O)C(C)(C)N=C1c1ccc(cn1)C#Cc1cccc(F)c1
InChI Key InChIKey=OEBGXOHGRFWELO-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 143693
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Rattus norvegicus (Rat))
Hoffmann-La Roche
US Patent
Hoffmann-La Roche
US Patent
Affinity DataKi: 18nMAssay Description:The pharmacological activity of the compounds was tested using the following method: cDNA encoding rat mGlu 5a receptor was transiently transfected i...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:cDNA encoding rat mGlu 5a receptor was transiently transfected into EBNA cells using a procedure described by E.-J. Schlaeger and K. Christensen (Cyt...More data for this Ligand-Target Pair