BDBM150751 CPR005231 (6)
SMILES COc1cc(ccc1O)-c1ccc2ccc(-c3cccc(c3)C(=O)NCCN(C)C)n2n1
InChI Key InChIKey=MCIDHQCNUZBVQJ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 150751
Affinity DataIC50: 247nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
Affinity DataKd: 240nMpH: 7.5Assay Description:40 µL of a solution containing 350-500 µM of CPR005231 (compound 6) were titrated into the 200 µL sample cell containing 25-55 µM DAPK1 (AA 1-285) or...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair