BDBM167418 US9073893, 16
SMILES NC(=O)c1cccc2[nH]n(C3CCN(CC3)C3CCC3)c(=O)c12
InChI Key InChIKey=VPFGQWNBEHLGLL-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 167418
Affinity DataIC50: 2.50E+3nMT: 2°CAssay Description:Cellular activity of PARP-1 inhibitors was assessed by measuring the inhibition of the hydrogen peroxide induced PAR formation in HeLa cells (ECACC)....More data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Affinity evaluation of the tested compounds and their selectivity with respect to the different PARP isoforms of interest was assessed in a displacem...More data for this Ligand-Target Pair