BDBM176591 US9120761, 5
SMILES COc1cc(ccc1Nc1ncc(c(CCc2cccc(c2)C(N)=O)n1)C(F)(F)F)C1CCNCC1
InChI Key InChIKey=UKXVRLBNBZAAIX-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 176591
TargetVascular endothelial growth factor receptor 3 [818-948,1003-1077](Homo sapiens (Human))
Cancer Therapeutics Crc
US Patent
Cancer Therapeutics Crc
US Patent
Affinity DataIC50: 5.75E+3nMpH: 7.4Assay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A biotin labeled peptide is used as substrate (amino acid sequ...More data for this Ligand-Target Pair
Affinity DataIC50: 7.20nMpH: 7.4Assay Description:A biotin labeled peptide is used as substrate (amino acid sequence: Biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2) S...More data for this Ligand-Target Pair