BDBM176593 US9120761, 7
SMILES CCN1CCC(CC1)c1ccc(Nc2ncc(c(Cc3ccccc3C(N)=O)n2)C(F)(F)F)c(OC)c1
InChI Key InChIKey=OVSGTWVJEXAGQC-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 176593
TargetVascular endothelial growth factor receptor 3 [818-948,1003-1077](Homo sapiens (Human))
Cancer Therapeutics Crc
US Patent
Cancer Therapeutics Crc
US Patent
Affinity DataIC50: 1.33E+4nMpH: 7.4Assay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A biotin labeled peptide is used as substrate (amino acid sequ...More data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMpH: 7.4Assay Description:A biotin labeled peptide is used as substrate (amino acid sequence: Biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2) S...More data for this Ligand-Target Pair