BDBM177913 US9120797, 11::US9120797, 12
SMILES CN(C)C1(CCC2(CC1)N(CCc1c2[nH]c2ccccc12)C(C)=O)c1ccccc1
InChI Key InChIKey=OZMIXURVHNPRPT-UHFFFAOYSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 177913
Affinity DataKi: 2.20nM ΔG°: -11.8kcal/moleT: 2°CAssay Description:The receptor affinity for the human mu-opiate receptor was determined in a homogeneous batch in microtitre plates. For this, dilution series of the p...More data for this Ligand-Target Pair
Affinity DataKi: 2.40nM ΔG°: -11.8kcal/molepH: 7.4 T: 2°CAssay Description:The cyclohexane derivatives of the general formula I were investigated in a receptor binding assay with 3H-nociceptin/orphanin FQ with membranes from...More data for this Ligand-Target Pair
Affinity DataKi: 2.90nM ΔG°: -11.6kcal/molepH: 7.4 T: 2°CAssay Description:The cyclohexane derivatives of the general formula I were investigated in a receptor binding assay with 3H-nociceptin/orphanin FQ with membranes from...More data for this Ligand-Target Pair
Affinity DataKi: 4.40nM ΔG°: -11.4kcal/moleT: 2°CAssay Description:The receptor affinity for the human mu-opiate receptor was determined in a homogeneous batch in microtitre plates. For this, dilution series of the p...More data for this Ligand-Target Pair