BDBM181014 US9133197, 6
SMILES CCCC(=O)c1nc(N)c2nc(-n3nccn3)n(C)c2n1
InChI Key InChIKey=DCITZRYVYKMQQH-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 181014
TargetAdenosine receptor A2a(Homo sapiens (Human))
Sigma-Tau Industrie Farmaceutiche Riunite
US Patent
Sigma-Tau Industrie Farmaceutiche Riunite
US Patent
Affinity DataKi: 19nMpH: 7.4Assay Description:The protein concentration of membrane suspension was determined using the Bradford method (Pierce, Rockford, Ill., USA) with bovine albumin as standa...More data for this Ligand-Target Pair
Affinity DataKi: 216nM ΔG°: -9.09kcal/molepH: 7.4 T: 2°CAssay Description:Competition binding experiments have been performed incubating membranes from CHO-K1 cells stably transfected with the human adenosine A1 receptor (c...More data for this Ligand-Target Pair