BDBM200906 US9233946, 5
SMILES CC(C)c1ccc2sc(c(C)c2c1)S(=O)(=O)Nc1cccc(c1)C(O)=O
InChI Key InChIKey=GMPUAEBALQTUPO-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 200906
Affinity DataIC50: 30nMAssay Description:Method A: The kinase activity of the bi-functional enzyme is readily quantified based on the production of F-2,6-P2 as described by Van Schaftingen e...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of PFKFB3 in human PANC-1 cells assessed as reduction in Fructose-2,6-Bisphosphate productionMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of PFKFB3 (unknown origin) by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Method B: The kinase activity of the bi-functional enzyme is readily quantified based on the production of ADP and F-2,6-P2 from ATP and F6P. The ADP...More data for this Ligand-Target Pair