BDBM20158 1-benzyl-3-[(4-chlorophenyl)amino]-4-phenyl-2,5-dihydro-1H-pyrrole-2,5-dione::GSK3987 Analogue::Substituted Maleimide, 6

SMILES Clc1ccc(NC2=C(C(=O)N(Cc3ccccc3)C2=O)c2ccccc2)cc1

InChI Key InChIKey=XNAXKONPRDDOBL-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 20158   

TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Glaxosmithkline

LigandPNGBDBM20158(1-benzyl-3-[(4-chlorophenyl)amino]-4-phenyl-2,5-di...)
Affinity DataEC50:  110nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Glaxosmithkline

LigandPNGBDBM20158(1-benzyl-3-[(4-chlorophenyl)amino]-4-phenyl-2,5-di...)
Affinity DataEC50:  130nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed