BDBM212436 JMV 3002::N-[1-[4-[(2,4-dimethoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
SMILES COc1ccc(Cn2c(CCc3ccccc3)nnc2C(Cc2c[nH]c3ccccc23)NC(=O)c2ccccn2)c(OC)c1
InChI Key InChIKey=UMGBPWZCCHVQAY-UHFFFAOYSA-N
Data 5 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 212436
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Homo sapiens (Human))
Université Montpellier 1
Université Montpellier 1
Affinity DataKi: 8.70nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
TargetDimer of Growth hormone secretagogue receptor type 1(Homo sapiens (Human))
Université Montpellier 1
Université Montpellier 1
Affinity DataKi: 9.90nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1/Isoform 1B of Growth hormone secretagogue receptor type 1 (1B)(Homo sapiens (Human))
Université Montpellier 1
Université Montpellier 1
Affinity DataKi: 19.3nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Homo sapiens (Human))
Université Montpellier 1
Université Montpellier 1
Affinity DataKi: 993nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair