BDBM224618 US9326978, 31
SMILES Cc1ccc(Nc2nc3ccccc3c3[nH]c(nc23)C2CCCC2)cc1
InChI Key InChIKey=FHLIAQGQHFKJLO-UHFFFAOYSA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 224618
TargetAdenosine receptor A3(Homo sapiens (Human))
The United States of America, Represented By The Secretary, Dept. of Health and Human Services
US Patent
The United States of America, Represented By The Secretary, Dept. of Health and Human Services
US Patent
Affinity DataKi: 1.19E+3nMpH: 8.0Assay Description:Each tube in the competitive binding assay contained 100 μl membrane suspension (20 μg protein), 50 μl [125I]-AB-MECA (0.5 nM), and 50...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
The United States of America, Represented By The Secretary, Dept. of Health and Human Services
US Patent
The United States of America, Represented By The Secretary, Dept. of Health and Human Services
US Patent
Affinity DataKi: 3.85E+3nMpH: 7.4Assay Description:For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
The United States of America, Represented By The Secretary, Dept. of Health and Human Services
US Patent
The United States of America, Represented By The Secretary, Dept. of Health and Human Services
US Patent
Affinity DataKi: 5.22E+3nMpH: 7.4Assay Description:For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°...More data for this Ligand-Target Pair