BDBM234859 US9353116, 18
SMILES COc1cc2ncnc(Nc3cccc(NC(=O)C=C)c3)c2cc1OC
InChI Key InChIKey=DBBOSESLOUEALZ-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 234859
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of The University of California
US Patent
The Regents of The University of California
US Patent
Affinity DataIC50: 1.66E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of The University of California
US Patent
The Regents of The University of California
US Patent
Affinity DataIC50: >5.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair