BDBM263493 (s)-2-(5-methoxy-4-oxobenzo[d][1,2,3]triazin-3 (4h)-yl)-n-(1-(4-(trifluoromethyl)phenyl)ethyl)acetamide::US10561662, Example 61::US11173161, EX 61::US9556130, test 61
SMILES COc1cccc2nnn(CC(=O)N[C@@H](C)c3ccc(cc3)C(F)(F)F)c(=O)c12
InChI Key InChIKey=TXINLWSEWPZSAH-NSHDSACASA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 263493
Affinity DataKi: 26nM ΔG°: -9.61kcal/molepH: 7.4 T: 2°CAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Membranes were removed from −80° C., thawed and diluted in cold radioligand assay buffer (20 mM HEPES pH 7.4/5 mM MgCl2/1 mM CaCl2/Roche protea...More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair