BDBM271163 7-(4-chloro-2-fluorobenzenesulfonyl)-2-methyl-4-[(2S)-2-(trifluoromethyl)morpholin-4-yl]-5H-pyrrolo[3,2-d]pyrimidin-6-amine::US10059713, Example 284

SMILES Cc1nc(N2CCO[C@@H](C2)C(F)(F)F)c2[nH]c(N)c(c2n1)S(=O)(=O)c1ccc(Cl)cc1F

InChI Key

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 271163   

TargetFree fatty acid receptor 2(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM271163(7-(4-chloro-2-fluorobenzenesulfonyl)-2-methyl-4-[(...)
Affinity DataEC50:  1nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent