BDBM27573 5-({3-[(methylamino)methyl]-1H-indazol-4-yl}oxy)benzene-1,3-dicarbonitrile::Indazole Derivative, 3

SMILES CNCc1n[nH]c2cccc(Oc3cc(cc(c3)C#N)C#N)c12

InChI Key InChIKey=GRLLIRKDPSDACJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 27573   

TargetGag-Pol polyprotein [588-1027](Human immunodeficiency virus type 1 group M subtyp...)
Pfizer

LigandPNGBDBM27573(5-({3-[(methylamino)methyl]-1H-indazol-4-yl}oxy)be...)
Affinity DataIC50: >3.00E+4nMpH: 7.8 T: 2°CAssay Description:The inhibition of the RNA-dependent DNA polymerase activity of the HIV-1 reverse transcriptase enzyme was measured using a primer extension assay. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed