BDBM275813 5-chloro-4-(5-chloro- 6-(2,2,3,3-tetrafluoro- propoxy)pyridin-3- yloxy)-N-(N,N- dimethylsulfamoyl)- 2-fluorobenzamide::US10071957, Example 30
SMILES CN(C)S(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(OCC(F)(F)C(F)F)c(Cl)c2)cc1F
InChI Key InChIKey=UOURQUTWYWICIZ-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 275813
Affinity DataIC50: 47.8nMpH: 7.4 T: 2°CAssay Description:Preparation of membranes containing recombinantly expressed sodium channels: Frozen recombinant cell pellets were thawed on ice and diluted to 4 time...More data for this Ligand-Target Pair
Affinity DataIC50: 34nMpH: 7.2Assay Description:Patch voltage clamp electrophysiology allows for the direct measurement and quantification of block of voltage-gated sodium channels (NaV's), and...More data for this Ligand-Target Pair