BDBM28129 4-[(2S)-2-{[(3S)-1-({[(1S)-1-(benzylcarbamoyl)-3-carbamoylpropyl]carbamoyl}methyl)-2-oxopiperidin-3-yl]carbamoyl}-2-{[(benzyloxy)carbonyl]amino}ethyl]phenoxyphosphonic acid::Freidinger lactam peptidomimetic, 2
SMILES NC(=O)CC[C@H](NC(=O)CN1CCC[C@H](NC(=O)[C@H](Cc2ccc(OP(O)(O)=O)cc2)NC(=O)OCc2ccccc2)C1=O)C(=O)NCc1ccccc1
InChI Key InChIKey=XKKAFDDGPKIMCW-DTXPUJKBSA-N
Data 1 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 28129
TargetSignal transducer and activator of transcription 3 [127-722](Mus musculus (mouse))
University of Michigan At Ann Arbor
University of Michigan At Ann Arbor
Affinity DataKi: 3.13E+3nM ΔG°: -7.43kcal/molepH: 7.5 T: 2°CAssay Description:The assay was based on the fluorescence polarization of the unbound small binding partner will be low, and its binding to a larger binding partner wi...More data for this Ligand-Target Pair