BDBM283134 4-[2-(4-amino-piperidin-1-yl)-5- (6-methoxypyridin-3-yl)-1-methyl- 6-oxo-1,6-dihydro-pyrimidin-4-yl]- benzonitrile::US10023543, Example 3::US10207999, Example 3::US10328077, Example 3::US10548896, Example 3::US10849898, Example 3::US10960005, Example 3::US11084793, Example 3::US9573930, Example 3::US9771329, Example 3::US9776974, Example 3
SMILES COc1ccc(cn1)-c1c(nc(N2CCC(N)CC2)n(C)c1=O)-c1ccc(cc1)C#N
InChI Key InChIKey=MJQRQURVBRMRKC-UHFFFAOYSA-N
Data 12 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 283134
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Celgene Quanticel Research
US Patent
Affinity DataIC50: <100nMAssay Description:This assay determines the ability of a test compound to inhibit LSD-1 demethylase activity. E. coli expressed full-length human LSD-1 (Accession numb...More data for this Ligand-Target Pair