BDBM283758 N-(4-(azetidin-3-ylidenemethyl)-3,5-difluorophenyl)-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide::US10023559, Example 83
SMILES CCc1n[nH]c(C(=O)Nc2cc(F)c(C=C3CNC3)c(F)c2)c1C
InChI Key InChIKey=UXYBPJXHXJWOHR-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 283758
Affinity DataKi: 0.900nMpH: 7.4Assay Description:HEK-293 cells stably expressing rat TAAR1 were maintained at 37° C. and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, heat in...More data for this Ligand-Target Pair
Affinity DatapH: 7.4Assay Description:HEK-293 cells stably expressing mouse TAAR1 were maintained at 37° C. and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, heat ...More data for this Ligand-Target Pair