BDBM289509 5-(2-isopropyl-1-(3-(4- methylpiperazin-1-yl)- bicyclo[1.1.1]pentan-1- yl)-1H-imidazol-4-yl)- 3-(trifluoromethoxy)- pyridin-2-amine::US10093664, Example 74
SMILES CC(C)c1nc(cn1C12CC(C1)(C2)N1CCN(C)CC1)-c1cnc(N)c(OC(F)(F)F)c1
InChI Key InChIKey=BTLRWVSEIUQULA-UHFFFAOYSA-N
Data 1 Kd
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 289509
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 4.5nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair