BDBM299125 2,2-difluoro-3- ((6S,8R)-6-(4-(2- (3-(fluoromethyl) azetidin-1- yl)ethoxy)-2- methoxyphenyl)- 8-methyl-3,6,8,9- tetrahydro-7H- pyrazolo[4,3- f]isoquinolin-7- yl)propan-1-ol::US10125135, Example 14
SMILES COc1cc(OCCN2CC(CF)C2)ccc1[C@H]1N(CC(F)(F)CO)[C@H](C)Cc2c1ccc1[nH]ncc21
InChI Key
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 299125
Affinity DataIC50: 3.5nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair