BDBM299150 2-((6S,8R)-7-((1- fluorocyclo- propyl)methyl)- 8-methyl-6,7,8,9- tetrahydro-3H- pyrazolo[4,3- f]isoquinolin-6- yl)-5-(2-(3- (fluoromethyl) azetidin-1- yl)ethoxy) benzonitrile::US10125135, Example 39
SMILES C[C@@H]1Cc2c(ccc3[nH]ncc23)[C@H](N1CC1(F)CC1)c1ccc(OCCN2CC(CF)C2)cc1C#N
InChI Key
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 299150
Affinity DataIC50: 2.80nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair