BDBM304009 US10138242, Compound 98
SMILES COc1ccc(CN2CCc3c(C2)c(nn3CCNC(C)C)C(=O)NCc2cccc3ccccc23)c2ccccc12
InChI Key InChIKey=KTVWXYGBCPXDAK-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 304009
Affinity DataEC50: 2.27E+3nMAssay Description:The assay uses two types of beads: donor beads are coupled with streptavidin, and acceptor beads are coupled with an anti His-tag antibody. Upon exci...More data for this Ligand-Target Pair
TargetPeroxisomal membrane protein PEX14(Homo sapiens (Human))
Technische Universit£T M£Nchen
Curated by ChEMBL
Technische Universit£T M£Nchen
Curated by ChEMBL
Affinity DataEC50: 7.89E+3nMAssay Description:Inhibition of biotinylated PEX5-derived ALSENWAQEFLA binding to human N-terminal His-tagged PEX14 (21 to 84 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strainżLister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair