BDBM310235 US10150760, Example 22.0::US10150760, Example 23.0

SMILES C[C@@H]([C@H](C)S(=O)(=O)Nc1nnc([C@@H]2CCCOC2)n1-c1c(F)cccc1F)c1ncc(C)cn1

InChI Key InChIKey=RQOBXESUTNRCQA-HRCADAONSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 310235   

TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM310235(US10150760, Example 22.0 | US10150760, Example 23....)
Affinity DataEC50:  110nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM310235(US10150760, Example 22.0 | US10150760, Example 23....)
Affinity DataEC50:  260nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent