BDBM321473 3-(6-(2-cyclopropylethyl)-2-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)-N,N-dimethylbenzamide::US10183009, Example 85

SMILES CN(C)C(=O)c1cccc(c1)-c1cn(CCC2CC2)c(=O)c2[nH]c(C)cc12

InChI Key InChIKey=UEWBABOUVBWVHO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 321473   

TargetChromatin remodeling regulator CECR2 [424-538](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM321473(3-(6-(2-cyclopropylethyl)-2-methyl-7-oxo-6,7-dihyd...)
Affinity DataIC50:  480nMAssay Description:His/Flag epitope tagged TAF1-BD21504-1635 was cloned, expressed, and purified to homogeneity. TAF1-BD2 binding and inhibition was assessed by monitor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent