BDBM346983 US10202379, Reference Example 724

SMILES CCc1cccc2CSc3c(F)cccc3[C@@H](N3CN([C@H](C)C(F)(F)F)C(=O)c4c(O)c(=O)ccn34)c12

InChI Key InChIKey=PMEODFRRPNLIRU-SPLOXXLWSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 346983   

TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM346983(US10202379, Reference Example 724)
Affinity DataEC50:  6.33nMAssay Description:A test sample was diluted with a culture medium to an appropriate concentration in advance, and then 2 to 5-fold serial dilution on a 96 well plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM346983(US10202379, Reference Example 724)
Affinity DataIC50:  5.07nMAssay Description:A test sample was diluted with a culture medium to an appropriate concentration in advance, and then 2 to 5-fold serial dilution on a 96 well plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent