BDBM371542 4-chloro-5-(((3R,5S)-1,5-dimethylpiperidin-3-yl)amino)-2-methylpyridazin-3(2H)-one::US10239861, Example 22
SMILES C[C@H]1C[C@H](CN(C)C1)Nc1cnn(C)c(=O)c1Cl
InChI Key InChIKey=MRZBXPNVEWAIIA-DTWKUNHWSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 371542
Affinity DataIC50: 21.5nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair