BDBM381334 4-Chloro-3-methyl-1-(tetrahydro- pyran-4-yl)-1H-pyrazolo[3,4- b]pyridine-5-carboxylic acid (4- chloro-phenyl)-amide::US10272074, Example 167
SMILES Cc1nn(C2CCOCC2)c2ncc(C(=O)Nc3ccc(Cl)cc3)c(Cl)c12
InChI Key InChIKey=RBRGBORCJQMFBD-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 381334
TargetGlucocorticoid receptor(Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute
US Patent
Sanford Burnham Prebys Medical Discovery Institute
US Patent
Affinity DataIC50: <50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair