BDBM381335 4-Chloro-3-methyl-1-(tetrahydro- pyran-4-yl)-1H-pyrazolo[3,4- b]pyridine-5-carboxylic acid (4- isopropyl-phenyl)-amide::US10272074, Example 168
SMILES CC(C)c1ccc(NC(=O)c2cnc3n(nc(C)c3c2Cl)C2CCOCC2)cc1
InChI Key InChIKey=VPWRKLYPONGENE-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 381335
TargetGlucocorticoid receptor(Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute
US Patent
Sanford Burnham Prebys Medical Discovery Institute
US Patent
Affinity DataIC50: <50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair