BDBM381439 4-chloro-N-(4-chlorophenyl)-1-((1- ethyl-1H-imidazol-2-yl)methyl)-3- methyl-1H-pyrazolo[3,4- b]pyridine-5-carboxamide::US10272074, Example 272
SMILES CCn1ccnc1Cn1nc(C)c2c(Cl)c(cnc12)C(=O)Nc1ccc(Cl)cc1
InChI Key InChIKey=XSQXKVLYMWGHFR-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 381439
TargetGlucocorticoid receptor(Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute
US Patent
Sanford Burnham Prebys Medical Discovery Institute
US Patent
Affinity DataIC50: <50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair