BDBM384295 Cis-2-(((2′-fluoro-5′-phenoxy-[1,1′-biphenyl]-4-yl)oxy)methyl)cyclopropanecarboxylic acid (racemate)::US9938222, Example 4::US9938222, Example 5

SMILES OC(=O)[C@@H]1C[C@@H]1COc1ccc(cc1)-c1cc(Oc2ccccc2)ccc1F

InChI Key InChIKey=AJTGGQOMNOFFQJ-IIBYNOLFSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 384295   

TargetFree fatty acid receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384295(Cis-2-(((2′-fluoro-5′-phenoxy-[1,1R...)
Affinity DataEC50:  2.11E+3nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384295(Cis-2-(((2′-fluoro-5′-phenoxy-[1,1R...)
Affinity DataEC50:  470nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent