BDBM384305 (Trans)-(+/−)-2-(((2′,3-difluoro-5′-phenoxy-[1,1′-biphenyl]-4-yl)oxy)methyl) cyclopropanecarboxylic acid::US9938222, Example 11::US9938222, Example 9

SMILES OC(=O)[C@H]1C[C@@H]1COc1ccc(cc1F)-c1cc(Oc2ccccc2)ccc1F

InChI Key InChIKey=CQUXGJOLCIJOLT-BEFAXECRSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 384305   

TargetFree fatty acid receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384305((Trans)-(+/−)-2-(((2′,3-difluoro-5R...)
Affinity DataEC50:  160nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384305((Trans)-(+/−)-2-(((2′,3-difluoro-5R...)
Affinity DataEC50:  80nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent