BDBM385711 4-(7-{[(4- fluorophenyl) methyl]amino}- [1,2,4]triazolo[1,5- a]pyridin-5- yl)benzonitrile::US10287286, Example 117

SMILES Fc1ccc(CNc2cc(-c3ccc(cc3)C#N)n3ncnc3c2)cc1

InChI Key InChIKey=DDBNRFRBPGDKLB-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 385711   

TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM385711(4-(7-{[(4- fluorophenyl) methyl]amino}- [1,2,4]tri...)
Affinity DataIC50:  5nMAssay Description:The IC50 values for the PHD1 enzyme (residues 1-407) were determined by mixing increasing amounts of a compound of the invention with a fixed amount ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent