BDBM385721 2-fluoro-4-{7- [(3,3,3- trifluoropropyl)- amino][1,2,4] triazolo- [1,5-a]pyridin-5- yl}benzonitrile::US10287286, Example 126

SMILES Fc1cc(ccc1C#N)-c1cc(NCCC(F)(F)F)cc2ncnn12

InChI Key InChIKey=VGCGIXOMVFHOFE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 385721   

TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM385721(2-fluoro-4-{7- [(3,3,3- trifluoropropyl)- amino][1...)
Affinity DataIC50:  53nMAssay Description:The IC50 values for the PHD1 enzyme (residues 1-407) were determined by mixing increasing amounts of a compound of the invention with a fixed amount ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent