BDBM385766 N-[5-(4-cyano-3- fluorophenyl)- [1,2,4]triazolo[1,5- a]pyridin-5-yl]-2- cyclopropyl- acetamide::US10287286, Example 169

SMILES Fc1cc(ccc1C#N)-c1cc(NC(=O)CC2CC2)cc2ncnn12

InChI Key InChIKey=UHZBVANUVKROCY-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 385766   

TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM385766(N-[5-(4-cyano-3- fluorophenyl)- [1,2,4]triazolo[1,...)
Affinity DataIC50:  49nMAssay Description:The IC50 values for the PHD1 enzyme (residues 1-407) were determined by mixing increasing amounts of a compound of the invention with a fixed amount ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent