BDBM403686 (1S,2S)-2-(4-((+/−)-3-Phenoxycyclohexyl)phenethyl)cyclopropanecarboxylic acid (cis-1,3-cyclohexyl isomer; Absolute Stereochemistry of the Cyclohexyl Moiety is Arbitrarily Drawn)::US10336684, Example 11::US10336684, Example 7::US10336684, Example 9

SMILES OC(=O)[C@H]1C[C@@H]1CCc1ccc(cc1)[C@@H]1CCC[C@@H](C1)Oc1ccccc1

InChI Key InChIKey=PBTFSZHZBADCEX-VAPSRWTKSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 403686   

TargetFree fatty acid receptor 4(Homo sapiens (Human))
Bristol=Myers Squibb

US Patent
LigandPNGBDBM403686((1S,2S)-2-(4-((+/−)-3-Phenoxycyclohexyl)phen...)
Affinity DataEC50:  920nMAssay Description:The human and mouse GPR120-mediated intracellular phosphorylated ERK assays were also established using CHO-K1 cells stably transfected with the shor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Bristol=Myers Squibb

US Patent
LigandPNGBDBM403686((1S,2S)-2-(4-((+/−)-3-Phenoxycyclohexyl)phen...)
Affinity DataEC50:  600nMAssay Description:The human and mouse GPR120-mediated intracellular phosphorylated ERK assays were also established using CHO-K1 cells stably transfected with the shor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Bristol=Myers Squibb

US Patent
LigandPNGBDBM403686((1S,2S)-2-(4-((+/−)-3-Phenoxycyclohexyl)phen...)
Affinity DataEC50:  650nMAssay Description:The human and mouse GPR120-mediated intracellular phosphorylated ERK assays were also established using CHO-K1 cells stably transfected with the shor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent