BDBM405072 1-[2-fluoro-4-(4-{2-[2-fluoro-5- (trifluoromethoxy)phenyl]acetamido}- 1H-1,2,3-triazol-1-yl)butyl]-N-{[3- (trifluoromethoxy)phenyl]methyl}- 1H-1,2,3-triazole-4-carboxamide::US10344025, Example 416::US11370786, Example 416
SMILES FC(CCn1cc(NC(=O)Cc2cc(OC(F)(F)F)ccc2F)nn1)Cn1cc(nn1)C(=O)NCc1cccc(OC(F)(F)F)c1
InChI Key InChIKey=YUADFEINGMENOR-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 405072
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Board of Regents, The University of Texas System
US Patent
Board of Regents, The University of Texas System
US Patent
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Board of Regents, The University of Texas System
US Patent
Board of Regents, The University of Texas System
US Patent
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair